摘要
本文报道了由1-对甲苯磺酰基4-氨基吲哚出发制得了五个创新霉素类化合物,精原细胞法实验表明,1-对甲苯磺酰基-3-三氟甲基创新霉素具有抗瘤活性。
This paper reported the synthesis of five analogues of Ch-uangxinmycin. It was shown that 1-Tosyl-3-trifluoro-methyl Chuangxin-mycin methyl ester exhibites antitumor activities by murine spermatogon-ial depletion assay.
出处
《中国抗生素杂志》
CAS
CSCD
北大核心
1992年第6期417-421,共5页
Chinese Journal of Antibiotics
关键词
创新霉素
抗瘤活性
Chuangxinmycin
l-Tosyl-3-trifluoro-methyl Chuangxin mycin
Antitumor activity