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20(S)-喜树碱及衍生物研究进展 被引量:1

Devolopment of the study on camptothecin and its derivatives
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出处 《西北药学杂志》 CAS 2001年第1期38-39,共2页 Northwest Pharmaceutical Journal
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同被引文献19

  • 1Van Ark-Otte J, Kedde MA, Van Der Vijgh WJF, et al. Determinants of CPT-11 and SN-38 activities in human lung cancer cells[J].Br J Cane, 1998, 77: 2171-2176.
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  • 3Danks MK, Morton CL, Krull EJ, et al. Comparison of activation of CPT-11 by rabbit and human carboxylesterases for use in enzyme/prodrug therapy[J]. Clin Canc Res, 1999,5:917-924.
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  • 6Iyer L, King CD. Genetic predisposition to the metabolism of irinotecan (CPT-11)[J]. J Clin Investig, 1998,101 : 847-854.
  • 7Monaghan G, Ryan M, Seddon R, et al. Genetic variation in bilirubin UDP-glucuronosyltrans-ferase gene promoter and Gilbert' s syndrome[J]. Lancet, 1996, 347 : 578-581.
  • 8Wasserman E, Myara A, Mick R, et al. Bilirubin (BIL) and SN-38: pharmacokinetic/pharmacodynamics correlation[J]. Ann Oncol, 1998,10:58.
  • 9Santos A, Zannetta S, Cresteil T, et al. Metabolism of irinotecan (CPT-11) by CYP3A4 and CYP3A5 in humans[J].Clin Cane Res, 2000,6:2012-2020.
  • 10Dodds HM, Haaz MC, Riou JF, et al. Identification of a new metabolite of CPT-11 (irinotecan) : pharmacological properties and activation to SN-38 [J]. J Pharmaeol Exp Ther, 1998,286: 578-583.

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