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替卡格雷合成路线图解 被引量:13

Graphical Synthetic Routes of Ticagrelor
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摘要 替卡格雷(ticagrelor,1),化学名为(1S,2S,3R,5S)-3-[7-[(1R,2S)-2-(3,4-二氟苯基)环丙胺基]-5-(丙硫基)-3H-[1,2,3]三唑[4,5-d]嘧啶-3-基]-5-(2-羟基乙氧基)环戊烷-1,2-二醇,由Astrazeneca公司研发,目前处于Ⅲ期临床研究。
出处 《中国医药工业杂志》 CAS CSCD 北大核心 2011年第2期146-150,149-150+148,共5页 Chinese Journal of Pharmaceuticals
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同被引文献84

  • 1张虹.邻二氟苯的合成与研究[J].有机氟工业,2006(3):14-16. 被引量:2
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  • 3Khile AS, Patel J, Trivedi N, et al. Improved processes for preparing ticagrelor intermediate, 4,6-dichloro-5-nitro-2- (propylthio) pyrimidine : WO, 2011101740 [P]. 2011-08-25.
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