摘要
综述了近年来阿朴菲类生物碱生物活性研究进展,包括肾上腺素受体作用活性、离子通道作用活性、抗血清素活性、细胞毒性、抗氧化活性、抗血小板聚集活性、神经系统活性、免疫调节活性、抗病毒活性以及其他活性等十个方面,并对其构效关系进行了初步分析。
Recent research on biological activities of aporphinoid alkaloids were reviewed, including adrenoceptor antagonistic effect, anfiserotonergic activity, ion chunnels blocking activity, cytotoxicity, antioxidative activity, anfiplatelet aggregation, effect on nervous system, immuno-mdulafion, antivirus activity and others. The structure-activity relationship was discussed briefly.
出处
《天然产物研究与开发》
CAS
CSCD
2006年第2期316-324,共9页
Natural Product Research and Development
关键词
阿朴菲类生物碱
生物活性
构效关系
进展
aporphinoid alkaloids
biological activities
stmcture-activity relationship
progress