A series of novel N-(4-(2-aryloxythiazol-5-yl)but-3-yn-2-yl)benzamide derivatives were designed and synthesized. Their structures were identified by IH NMR and elemental analyses. Preliminary bioassays indicated t...A series of novel N-(4-(2-aryloxythiazol-5-yl)but-3-yn-2-yl)benzamide derivatives were designed and synthesized. Their structures were identified by IH NMR and elemental analyses. Preliminary bioassays indicated that some title compounds provided 〉 80% control of Selerotinia selerotiorum at 50 μg/mL and 〉 70% herbicidal activities against B. campestris at 100 μg/mL. Their structure-activities relationships were also discussed.展开更多
基金We are grateful for financial support by the National Basic Research Program of China (973 Program),the National Natural Science Foundation of China,the National Key Technologies R&D Program
文摘A series of novel N-(4-(2-aryloxythiazol-5-yl)but-3-yn-2-yl)benzamide derivatives were designed and synthesized. Their structures were identified by IH NMR and elemental analyses. Preliminary bioassays indicated that some title compounds provided 〉 80% control of Selerotinia selerotiorum at 50 μg/mL and 〉 70% herbicidal activities against B. campestris at 100 μg/mL. Their structure-activities relationships were also discussed.