In view of potent antimicrobial and anti-inflammatory activities exhibited by S-substituted imidazolones, a variety of novel imidazolone analogs 3a-I were synthesized by the condensation of different substituted oxazo...In view of potent antimicrobial and anti-inflammatory activities exhibited by S-substituted imidazolones, a variety of novel imidazolone analogs 3a-I were synthesized by the condensation of different substituted oxazolones I with various aromatic amines 2. All the synthesized compounds were screened for in vitro activities against a panel of Gram-positive and Gram-negative bacteria and the yeast-like pathogenic fungus Candida albicans. Several analogs produced good or moderate activities particularly against the tested Gram-positive bacteria Micrococcus luteus and Gram-negative bacteria Pseudornonas aeruginosa and, Meanwhile, compounds 3b and 3c displayed marked antifungal activity against C. albicans. In addition, the in vivo anti-inflammatory activity of the synthesized compounds was determined using the carrageenin-induced paw oedema method in rats. Two of S-substituted imidazo/one derivatives, 3k and 3d show good anti-inflammatory activity. The structures of all the newly svnthesized compounds were elucidated using IR, 1H NMR and 13C NMR.展开更多
Greenhouse technology is a practical option for the production and drying of agricultural products in controlled environment. For the successful design of a greenhouse, the selection of a suitable shape and orientatio...Greenhouse technology is a practical option for the production and drying of agricultural products in controlled environment. For the successful design of a greenhouse, the selection of a suitable shape and orientation is of great importance. Of various shapes of greenhouses, the even-span roof and the Quonset shape greenhouses are the most commonly used for crop cultivation and drying. The orientation of greenhouses is kept east-west for maximum utilization of solar radiations. Hybrid and modified greenhouse dryers have been proposed for drying of products. The agricultural products dried in greenhouses are found to be better in quality as compared to open sun drying because they are protected from dust, rain, insects, birds and animals. Moreover, various greenhouses shapes along with their applications have been reviewed.展开更多
文摘In view of potent antimicrobial and anti-inflammatory activities exhibited by S-substituted imidazolones, a variety of novel imidazolone analogs 3a-I were synthesized by the condensation of different substituted oxazolones I with various aromatic amines 2. All the synthesized compounds were screened for in vitro activities against a panel of Gram-positive and Gram-negative bacteria and the yeast-like pathogenic fungus Candida albicans. Several analogs produced good or moderate activities particularly against the tested Gram-positive bacteria Micrococcus luteus and Gram-negative bacteria Pseudornonas aeruginosa and, Meanwhile, compounds 3b and 3c displayed marked antifungal activity against C. albicans. In addition, the in vivo anti-inflammatory activity of the synthesized compounds was determined using the carrageenin-induced paw oedema method in rats. Two of S-substituted imidazo/one derivatives, 3k and 3d show good anti-inflammatory activity. The structures of all the newly svnthesized compounds were elucidated using IR, 1H NMR and 13C NMR.
文摘Greenhouse technology is a practical option for the production and drying of agricultural products in controlled environment. For the successful design of a greenhouse, the selection of a suitable shape and orientation is of great importance. Of various shapes of greenhouses, the even-span roof and the Quonset shape greenhouses are the most commonly used for crop cultivation and drying. The orientation of greenhouses is kept east-west for maximum utilization of solar radiations. Hybrid and modified greenhouse dryers have been proposed for drying of products. The agricultural products dried in greenhouses are found to be better in quality as compared to open sun drying because they are protected from dust, rain, insects, birds and animals. Moreover, various greenhouses shapes along with their applications have been reviewed.
